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PreviewIssue dateOnline publication dateTitleAuthor(s)
saeed_mohamed_e._m.-drug_repurposi-20210510114527807.pdf.jpg202110-May-2021Drug repurposing using transcriptome sequencing and virtual drug screening in a patient with glioblastomaSaeed, Mohamed E. M.; Kadioglu, Onat; Greten, Henry Johannes; Yildirim, Adem; Mayr, Katharina; Wenz, Frederik; Giordano, Frank; Efferth, Thomas
barthels_fabian-banδit__b’-fac-20210628203840983.pdf.jpg202129-Jun-2021BANΔIT: B’-factor analysis for drug design and structural biologyBarthels, Fabian; Schirmeister, Tanja; Kersten, Christian
welker_armin-structure-acti-20210621155711267.pdf.jpg202128-Jun-2021Structure-activity relationships of benzamides and isoindolines designed as SARS-CoV protease inhibitors effective against SARS-CoV-2Welker, Armin; Kersten, Christian; Müller, Christin; Madhugiri, Ramakanth; Zimmer, Collin; Müller, Patrick; Zimmermann, Robert; Hammerschmidt, Stefan; Maus, Hannah; Ziebuhr, John; Sotriffer, Christoph; Schirmeister, Tanja
x-im30_idps_form-20210420093443760.pdf.jpg202023-Apr-2021IM30 IDPs form a membrane-protective carpet upon super-complex disassemblyJunglas, Benedikt; Orru, Roberto; Axt, Amelie; Siebenaller, Carmen; Steinchen, Wieland; Heidrich, Jennifer; Hellmich, Ute A.; Hellmann, Nadja; Wolf, Eva; Weber, Stefan A. L.; Schneider, Dirk
cymer_florian-small_residues-20211115121527126.pdf.jpg202115-Nov-2021Small residues inhibit homo-dimerization of the human carbonic anhydrase XII transmembrane domainCymer, Florian; Schneider, Dirk
barthels_fabian-asymmetric_dis-20210805114859449.pdf.jpg202013-Aug-2021Asymmetric disulfanylbenzamides as irreversible and selective inhibitors of Staphylococcus aureus sortase ABarthels, Fabian; Marincola, Gabriella; Marciniak, Tessa; Konhäuser, Matthias; Hammerschmidt, Stefan; Bierlmeier, Jan; Distler, Ute; Wich, Peter R.; Tenzer, Stefan; Schwarzer, Dirk; Ziebuhr, Wilma; Schirmeister, Tanja
wagener_karolin-targeting_of_i-20210812113737053.pdf.jpg202013-Aug-2021Targeting of immune cells with trimannosylated liposomesWagener, Karolin; Bros, Matthias; Krumb, Matthias; Langhanki, Jens; Pektor, Stefanie; Worm, Matthias; Schinnerer, Meike; Montermann, Evelyn; Miederer, Matthias; Frey, Holger; Opatz, Till; Rösch, Frank
stengelin_elena-bone_scaffolds-20210804000148620.pdf.jpg20209-Aug-2021Bone scaffolds based on degradable vaterite/PEG-composite microgelsStengelin, Elena; Kuzmina, Alena; Beltramo, Guillermo L.; Koziol, Martha F.; Besch, Laura; Schröder, Romina; Unger, Ronald E.; Tremel, Wolfgang; Seiffert, Sebastian
özenver_nadire-chemometric_an-20210209112718237.pdf.jpg20209-Feb-2021Chemometric and transcriptomic profiling, microtubule disruption and cell death induction by secalonic acid in tumor cellsÖzenver, Nadire; Dawood, Mona; Fleischer, Edmond; Klinger, Anette; Efferth, Thomas
kadioglu_onat-identification-20210209101413928.pdf.jpg20209-Feb-2021Identification of novel rare ABCC1 transporter mutations in tumor biopsies of cancer patientsKadioglu, Onat; Saeed, Mohamed; Munder, Markus; Spuller, Andreas; Greten, Henry Johannes; Efferth, Thomas