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PreviewIssue dateOnline publication dateTitleAuthor(s)
welker_armin-structure-acti-20210621155711267.pdf.jpg202128-Jun-2021Structure-activity relationships of benzamides and isoindolines designed as SARS-CoV protease inhibitors effective against SARS-CoV-2Welker, Armin; Kersten, Christian; Müller, Christin; Madhugiri, Ramakanth; Zimmer, Collin; Müller, Patrick; Zimmermann, Robert; Hammerschmidt, Stefan; Maus, Hannah; Ziebuhr, John; Sotriffer, Christoph; Schirmeister, Tanja
analysis_of_hyperforin_st_joh-20230118131954936.pdf.jpg202218-Jan-2023Analysis of hyperforin (St. John’s wort) action at TRPC6 channel leads to the development of a new class of antidepressant drugsEl Hamdaoui, Yamina; Zheng, Fang; Fritz, Nikolas; Ye, Lian; Tran, Mai Anh; Schwickert, Kevin; Schirmeister, Tanja; Braeuning, Albert; Lichtenstein, Dajana; Hellmich, Ute A.; Weikert, Dorothee; Heinrich, Markus; Treccani, Giulia; Schäfer, Michael K. E.; Nowak, Gabriel; Nürnberg, Bernd; Alzheimer, Christian; Müller, Christian P.; Friedland, Kristina
subnanomolar_cathepsin_s_inhi-20230901153132231.pdf.jpg202312-Sep-2023Subnanomolar cathepsin S inhibitors with high selectivity : optimizing covalent reversible α-fluorovinylsulfones and α-sulfonates as potential immunomodulators cancerFuchs, Natalie; Meta, Mergim; Lantzberg, Bellinda; Bros, Matthias; Kuan, Seah Ling; Weil, Tanja; Schirmeister, Tanja
2sulfonylpyrimidines_as_privi-20230302115838017.pdf.jpg20212-Mar-20232-sulfonylpyrimidines as privileged warheads for the development of S. aureus sortase A inhibitorsBarthels, Fabian; Meyr, Jessica; Hammerschmidt, Stefan J.; Marciniak, Tessa; Räder, Hans-Joachim; Ziebuhr, Wilma; Engels, Bernd; Schirmeister, Tanja
sarscovplproinhibitoren_als_m-20220701134011960.pdf.jpg20214-Jul-2022SARS-CoV-PLpro-Inhibitoren als mögliche Breitspektrum-VirostatikaHammerschmidt, Stefan Josef; Müller, Patrick; Schirmeister, Tanja
a_competition_smfret_assay_to-20240216093225346.pdf.jpg202316-Feb-2024A competition smFRET assay to study ligand-induced conformational changes of the dengue virus proteaseMaus, Hannah; Hinze, Gerald; Hammerschmidt, Stefan Josef; Basché, Thomas; Schirmeister, Tanja