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PreviewIssue dateOnline publication dateTitleAuthor(s)
sarscovplproinhibitoren_als_m-20220701134011960.pdf.jpg20214-Jul-2022SARS-CoV-PLpro-Inhibitoren als mögliche Breitspektrum-VirostatikaHammerschmidt, Stefan Josef; Müller, Patrick; Schirmeister, Tanja
59032.pdf.jpg201916-Apr-2019Natural product repertoire of the genus AmphimedonShady, Nourhan Hisham; Fouad, Mostafa A.; Kamel, Mohamed Salah; Schirmeister, Tanja; Abdelmohsen, Usama Ramadan
59874.pdf.jpg202023-Jun-2020Naphthoquinones as covalent reversible inhibitors of cysteine proteases : studies on inhibition mechanism and kineticsKlein, Philipp; Barthels, Fabian; Johe, Patrick; Wagner, Annika; Tenzer, Stefan; Distler, Ute; Le, Thien Anh; Schmid, Paul; Engel, Volker; Engels, Bernd; Hellmich, Ute; Opatz, Till; Schirmeister, Tanja
59826.pdf.jpg202018-May-2020New cysteine protease inhibitors : electrophilic (het)arenes and unexpected prodrug identification for the trypanosoma protease rhodesainKlein, Philipp; Johe, Patrick; Wagner, Annika; Jung, Sascha; Kühlborn, Jonas; Barthels, Fabian; Tenzer, Stefan; Distler, Ute; Waigel, Waldemar; Engels, Bernd; Hellmich, Ute; Opatz, Till; Schirmeister, Tanja
chemical_space_virtual_screen-20230418075719562.pdf.jpg202318-Apr-2023Chemical space virtual screening against hard-to-drug RNA methyltransferases DNMT2 and NSUN6Zimmermann, Robert A.; Fischer, Tim R.; Schwickert, Marvin; Nidoieva, Zarina; Schirmeister, Tanja; Kersten, Christian
2sulfonylpyrimidines_as_privi-20230302115838017.pdf.jpg20212-Mar-20232-sulfonylpyrimidines as privileged warheads for the development of S. aureus sortase A inhibitorsBarthels, Fabian; Meyr, Jessica; Hammerschmidt, Stefan J.; Marciniak, Tessa; Räder, Hans-Joachim; Ziebuhr, Wilma; Engels, Bernd; Schirmeister, Tanja
a_competition_smfret_assay_to-20240216093225346.pdf.jpg202316-Feb-2024A competition smFRET assay to study ligand-induced conformational changes of the dengue virus proteaseMaus, Hannah; Hinze, Gerald; Hammerschmidt, Stefan Josef; Basché, Thomas; Schirmeister, Tanja
ligandbased_design_of_selecti-20240315084304365.pdf.jpg202415-Mar-2024Ligand-based design of selective peptidomimetic uPA and TMPRSS2 inhibitors with arg bioisosteresMüller, Patrick; Zimmer, Collin; Frey, Ariane; Holzmann, Gideon; Weldert, Annabelle Carolin; Schirmeister, Tanja