A total synthesis of (−)-strychnine using photoredox catalysis

dc.contributor.authorWiechert, Rainer
dc.contributor.authorGeske, Leander
dc.contributor.authorHammes, Jasmin
dc.contributor.authorTuncer, Dogus
dc.contributor.authorOpatz, Till
dc.date.accessioned2026-08-04T13:51:54Z
dc.date.issued2026
dc.description.abstractA concise route toward (−)-strychnine is presented. Key steps include the photoredox-catalytic C2-cyanomethylation of Boc-l-Trp-OMe and a condensation-electrocyclization cascade linking two fragments convergently to obtain an advanced intermediate. A photochemical decarboxylation provided convenient access to strychnofluorine, which could be transformed through the Wieland–Gumlich aldehyde to strychnine. All building blocks can be traced back to renewable sources.en
dc.identifier.doihttps://doi.org/10.25358/openscience-16043
dc.identifier.urihttps://openscience.ub.uni-mainz.de/handle/20.500.12030/16064
dc.language.isoeng
dc.rightsCC-BY-4.0
dc.rights.urihttps://creativecommons.org/licenses/by/4.0/
dc.subject.ddc540 Chemiede
dc.subject.ddc540 Chemistry and allied sciencesen
dc.titleA total synthesis of (−)-strychnine using photoredox catalysisen
dc.typeZeitschriftenaufsatz
jgu.apc.netprice0,00
jgu.apc.price0,00
jgu.apc.taxrate0
jgu.apc.transformationcontractACS
jgu.dfg.year2026
jgu.identifier.uuid16d29412-770a-4d44-ac33-27327cb905ed
jgu.journal.issue3
jgu.journal.titleJACS Au : an open access journal of the American Chemical Society
jgu.journal.volume6
jgu.nationalcurrency.eur0,00
jgu.organisation.departmentFB 09 Chemie, Pharmazie u. Geowissensch.
jgu.organisation.nameJohannes Gutenberg-Universität Mainz
jgu.organisation.number7950
jgu.organisation.placeMainz
jgu.organisation.rorhttps://ror.org/023b0x485
jgu.pages.end1826
jgu.pages.start1822
jgu.publisher.doi10.1021/jacsau.5c01709
jgu.publisher.eissn2691-3704
jgu.publisher.nameACS
jgu.publisher.placeWashington, DC
jgu.publisher.year2026
jgu.rights.accessrightsopenAccess
jgu.subject.ddccode540
jgu.subject.dfgNaturwissenschaften
jgu.type.dinitypeArticleen_GB
jgu.type.resourceText
jgu.type.versionPublished version

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