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PreviewIssue dateOnline publication dateTitleAuthor(s)
59032.pdf.jpg201916-Apr-2019Natural product repertoire of the genus AmphimedonShady, Nourhan Hisham; Fouad, Mostafa A.; Kamel, Mohamed Salah; Schirmeister, Tanja; Abdelmohsen, Usama Ramadan
barthels_fabian-banδit__b’-fac-20210628203840983.pdf.jpg202129-Jun-2021BANΔIT: B’-factor analysis for drug design and structural biologyBarthels, Fabian; Schirmeister, Tanja; Kersten, Christian
barthels_fabian-asymmetric_dis-20210805114859449.pdf.jpg202013-Aug-2021Asymmetric disulfanylbenzamides as irreversible and selective inhibitors of Staphylococcus aureus sortase ABarthels, Fabian; Marincola, Gabriella; Marciniak, Tessa; Konhäuser, Matthias; Hammerschmidt, Stefan; Bierlmeier, Jan; Distler, Ute; Wich, Peter R.; Tenzer, Stefan; Schwarzer, Dirk; Ziebuhr, Wilma; Schirmeister, Tanja
cytotoxicity_of_endoperoxides-20220925182710959.pdf.jpg201721-Oct-2022Cytotoxicity of endoperoxides from the Caribbean sponge Plakortis halichondrioides towards sensitive and multidrug-resistant leukemia cells : acids vs. esters activity evaluationSchirmeister, Tanja; Oli, Swarna; Wu, Hongmei; Della Sala, Gerardo; Costantino, Valeria; Seo, Ean-Jeong; Efferth, Thomas
identification_of_plakortide_-20220510090302657.pdf.jpg201410-May-2022Identification of plakortide E from the Caribbean sponge Plakortis halichondroides as a trypanocidal protease inhibitor using bioactivity-guided fractionationOli, Swarna; Abdelmohsen, Usama Ramadan; Hentschel, Ute; Schirmeister, Tanja
welker_armin-structure-acti-20210621155711267.pdf.jpg202128-Jun-2021Structure-activity relationships of benzamides and isoindolines designed as SARS-CoV protease inhibitors effective against SARS-CoV-2Welker, Armin; Kersten, Christian; Müller, Christin; Madhugiri, Ramakanth; Zimmer, Collin; Müller, Patrick; Zimmermann, Robert; Hammerschmidt, Stefan; Maus, Hannah; Ziebuhr, John; Sotriffer, Christoph; Schirmeister, Tanja
novel_dengue_virus_ns2bns3_pr-20220913202020725.pdf.jpg20157-Dec-2022Novel dengue virus NS2B/NS3 protease inhibitorsWu, Hongmei; Bock, Stefanie; Snitko, Mariya; Berger, Thilo; Weidner, Thomas; Holloway, Steven; Kanitz, Manuel; Diederich, Wibke E.; Steuber, Holger; Walter, Christof; Hofmann, Daniela; Weißbrich, Benedikt; Spannaus, Ralf; Acosta, Eliana G.; Bartenschlager, Ralf; Engels, Bernd; Schirmeister, Tanja; Bodem, Jochen
59109.pdf.jpg201917-Jun-2019Identification of a potential allosteric site of Golgi α-mannosidase II using computer-aided drug designIrsheid, Lina; Wehler, Thomas; Borek, Christoph; Kiefer, Werner; Brenk, Ruth; Ortiz-Soto, Maria Elena; Seibel, Jürgen; Schirmeister, Tanja
59874.pdf.jpg202023-Jun-2020Naphthoquinones as covalent reversible inhibitors of cysteine proteases : studies on inhibition mechanism and kineticsKlein, Philipp; Barthels, Fabian; Johe, Patrick; Wagner, Annika; Tenzer, Stefan; Distler, Ute; Le, Thien Anh; Schmid, Paul; Engel, Volker; Engels, Bernd; Hellmich, Ute; Opatz, Till; Schirmeister, Tanja
59826.pdf.jpg202018-May-2020New cysteine protease inhibitors : electrophilic (het)arenes and unexpected prodrug identification for the trypanosoma protease rhodesainKlein, Philipp; Johe, Patrick; Wagner, Annika; Jung, Sascha; Kühlborn, Jonas; Barthels, Fabian; Tenzer, Stefan; Distler, Ute; Waigel, Waldemar; Engels, Bernd; Hellmich, Ute; Opatz, Till; Schirmeister, Tanja