Browsing by Author Schirmeister, Tanja

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ligandbased_design_of_selecti-20240315084304365.pdf.jpg202415-Mar-2024Ligand-based design of selective peptidomimetic uPA and TMPRSS2 inhibitors with arg bioisosteresMüller, Patrick; Zimmer, Collin; Frey, Ariane; Holzmann, Gideon; Weldert, Annabelle Carolin; Schirmeister, Tanja
59874.pdf.jpg202023-Jun-2020Naphthoquinones as covalent reversible inhibitors of cysteine proteases : studies on inhibition mechanism and kineticsKlein, Philipp; Barthels, Fabian; Johe, Patrick; Wagner, Annika; Tenzer, Stefan; Distler, Ute; Le, Thien Anh; Schmid, Paul; Engel, Volker; Engels, Bernd; Hellmich, Ute; Opatz, Till; Schirmeister, Tanja
59032.pdf.jpg201916-Apr-2019Natural product repertoire of the genus AmphimedonShady, Nourhan Hisham; Fouad, Mostafa A.; Kamel, Mohamed Salah; Schirmeister, Tanja; Abdelmohsen, Usama Ramadan
59826.pdf.jpg202018-May-2020New cysteine protease inhibitors : electrophilic (het)arenes and unexpected prodrug identification for the trypanosoma protease rhodesainKlein, Philipp; Johe, Patrick; Wagner, Annika; Jung, Sascha; Kühlborn, Jonas; Barthels, Fabian; Tenzer, Stefan; Distler, Ute; Waigel, Waldemar; Engels, Bernd; Hellmich, Ute; Opatz, Till; Schirmeister, Tanja
next_generation_of_fluorometr-20230914114142028.pdf.jpg202314-Sep-2023Next generation of fluorometric protease assays : 7-nitrobenz-2-oxa-1,3-diazol-4-yl-amides (NBD-amides) as class-spanning protease substratesMaus, Hannah; Müller, Patrick; Meta, Mergim; Hoba, Sabrina N.; Hammerschmidt, Stefan J.; Zimmermann, Robert A.; Zimmer, Collin; Fuchs, Natalie; Schirmeister, Tanja; Barthels, Fabian
novel_dengue_virus_ns2bns3_pr-20220913202020725.pdf.jpg20157-Dec-2022Novel dengue virus NS2B/NS3 protease inhibitorsWu, Hongmei; Bock, Stefanie; Snitko, Mariya; Berger, Thilo; Weidner, Thomas; Holloway, Steven; Kanitz, Manuel; Diederich, Wibke E.; Steuber, Holger; Walter, Christof; Hofmann, Daniela; Weißbrich, Benedikt; Spannaus, Ralf; Acosta, Eliana G.; Bartenschlager, Ralf; Engels, Bernd; Schirmeister, Tanja; Bodem, Jochen
sarscovplproinhibitoren_als_m-20220701134011960.pdf.jpg20214-Jul-2022SARS-CoV-PLpro-Inhibitoren als mögliche Breitspektrum-VirostatikaHammerschmidt, Stefan Josef; Müller, Patrick; Schirmeister, Tanja
welker_armin-structure-acti-20210621155711267.pdf.jpg202128-Jun-2021Structure-activity relationships of benzamides and isoindolines designed as SARS-CoV protease inhibitors effective against SARS-CoV-2Welker, Armin; Kersten, Christian; Müller, Christin; Madhugiri, Ramakanth; Zimmer, Collin; Müller, Patrick; Zimmermann, Robert; Hammerschmidt, Stefan; Maus, Hannah; Ziebuhr, John; Sotriffer, Christoph; Schirmeister, Tanja
subnanomolar_cathepsin_s_inhi-20230901153132231.pdf.jpg202312-Sep-2023Subnanomolar cathepsin S inhibitors with high selectivity : optimizing covalent reversible α-fluorovinylsulfones and α-sulfonates as potential immunomodulators cancerFuchs, Natalie; Meta, Mergim; Lantzberg, Bellinda; Bros, Matthias; Kuan, Seah Ling; Weil, Tanja; Schirmeister, Tanja